中间体API Intermediates

2019-07-01


■雷西纳得;lesnurad
878672-00-5Lesinurad  
878671-95-51-cyclopropyl-4-isothiocyanatonaphthalene 
878671-98-8methyl   2-((5-amino-4-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazol-3-yl)thio)acetate 
878671-96-63-amino-4-(4-cyclopropylnaphthalen-1-yl)-1H-1,2,4-triazole-5(4H)-thione 
1533519-92-44-cyclopropylnaphthalen-1-amine   HCl 
1533519-84-44-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazole-3-thiol 
■马西替坦;Macitentan
441798-33-0Macitentan 
706811-25-85-(4-bromophenyl)pyrimidine-4,6-diol 
146533-41-75-(4-bromophenyl)-4,6-dichloropyrimidine 
1878-68-84-Bromophenylacetic   acid 
149506-35-4Dimethyl   (4-Bromophenyl)-malonate 
1642873-03-7N-propylsulfamide   sodium salt 
■帕布昔利布;Palbociclib
571190-30-2Palbociclib
1016636-70-26-Bromo-2-chloro-8-cyclopentyl-5-methylpyrido[2,3-d]pyrimidin-7(8H)-one
571188-59-5tert-Butyl   4-(6-aminopyridin-3-yl)piperazine-1-carboxylate
■恩杂鲁胺;Enzalutamide
915087-33-1Enzalutamide
915087-24-0 2-fluoro-N-methyl-4-nitrobenzamide
915087-25-14-amino-2-fluoro-N-methylbenzamide 
143782-23-4 4-Isothiocyanato-2-(trifluoromethyl)benzonitrile 
915087-32-04-((2-cyanopropan-2-yl)amino)-2-fluoro-N-methylbenzamide
1289942-66-0 N-[3-Fluoro-4-[(methylamino)carbonyl]phenyl]-2-methylalanine
■鲁索利替尼; Ruxolitinib
941678-49-5Ruxolitinib
3680-69-14-chloro-7H-pyrrolo(2,3-d)Pyrimidine
269410-08-4Pyrazole-4-boronic   acid pinacol ester 
941685-27-44-(1H-pyrazol-4-yl)-7-((2-(trimethylsilyl)ethoxy)methyl)-7H-pyrrolo[2,3-d]pyrimidine
18997-19-8(4-chloro-7H-pyrrolo[2,3-d]pyrimidin-7-yl)methyl   pivalate
1029716-44-61-(1-ethoxyethyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole
 1146629-77-7(4-(1H-pyrazol-4-yl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)methyl   pivalate
591769-05-0(E)-3-cyclopentylacrylonitrile 
1236033-05-8(4-(1-(2-cyano-1-cyclopentylethyl)-1H-pyrazol-4-yl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)methyl   pivalate
■克唑替尼;Crizotinib
877399-52-5Crizotinib
330156-50-81.   (S)-1-(2,6-Dichloro-3-fluorophenyl)ethanol
877399-00-32.   (R)-5-bromo-3-[1-(2,6-dichloro-3-fluoropehnyl)ethoxy]pyridin-2-amine
877399-73-03.   4-(4-Iodo-pyrazol-1-yl)-piperidine-1-carboxylic acid tert-butyl ester
877399-74-14.   tert-Butyl   4-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]piperidine-1-carboxylate
■雷特格韦;Raltegravir
518048-05-0Raltegravir 
888504-27-61,6-dihydro-5-hydroxy-1-methyl-2-[1-methyl-1-[[(phenylmethoxy)carbonyl]amino]ethyl]-6-oxo-4-Pyrimidinecarboxylic   acid methyl ester 
519032-08-7 Methyl2-(1-{[(benzyloxy)carbonyl]aMino}-1-Methylethyl)-5,6-dihydroxypyriMidine-4-carboxyllate 
888504-28-7 5-Methyl-1,3,4-oxadiazole-2-carboxylic acid   potassium salt
518048-03-82-(1-Amino-1-methylethyl)-N-(4-fluorobenzyl)-5-hydroxy-1-methyl-6-oxo-1,6-dihydropyrimidine-4-carboxamide 
■鲁索曲波帕;Lusutrombopag
1110768-00-7Lusutrombopag
1110767-89-9(E)-3,5-dichloro-4-(3-ethoxy-2-methyl-3-oxoprop-1-enyl)benzoic   acid
1110767-98-0(S)-4-(3-(1-(hexyloxy)ethyl)-2-methoxyphenyl)thiazol-2-amine
■维拉帕尼;Veliparib
■依鲁替尼;Ibrutinib
936563-96-1Ibrutinib
 330786-24-8 1.   3-(4-Phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
143900-44-12.   (S)-1-Boc-3-hydroxypiperidine 
2380-63-43.   1H-pyrazolo[3,4-d]pyrimidin-4-amine 
1276110-38-34.   tert-butyl-(R)-3-(4-amino-3-iodo-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidine-1-   carboxylate 
■帕唑帕尼;Pazopanib
444731-52-6Pazopanib
3934-20-12,4-Dichloropyrimidine
6973-09-73-Amino-6-methylbenzenesulfonamide
635702-60-22,3-dimethyl-2H-indazol-6-amine   hydrochloride
■艾代拉里斯;Idelalisib
870281-82-6Idelalisib
870281-86-0(S)-2-(1-aminopropyl)-5-fluoro-3-phenylquinazolin-4(3H)-one
870281-85-9tert-butyl   (S)-(1-(5-fluoro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)propyl)carbamate
870281-84-8tert-butyl   (S)-(1-(2-fluoro-6-nitro-N-phenylbenzamido)-1-oxobutan-2-yl)carbamate
1417456-04-22-amino-6-fluoro-N-phenylbenzamide
■帕纳替尼;Ponatinib
943319-70-8Ponatinib
694499-26-84-(4-Methylpiperazinomethyl)-3-(trifluoromethyl)aniline 
943320-50-13-iodo-4-Methyl-N-(4-((4-Methylpiperazin-1-yl)Methyl)-3-(trifluoroMethyl)phenyl)benzaMide 
18087-73-53-BROMOIMIDAZO[1,2-B]PYRIDAZINE 
943320-61-43-Ethynylimidazo[1,2-b]pyridazine 
[66-55-2Imidazo[1,2-b]pyridazine
■克瑞沙硼;Crisaborole
906673-24-35-(4-cyanophenoxy)-2,3-dihydro-1-hydroxy-2,1-benzoxaborole
906673-45-84-[4-Bromo-3-(hydroxymethyl)   phenoxy]benzonitrile
906673-54-94-(4-Bromo-3-formylphenoxy)   benzonitrile
1160182-44-44-Bromo-3-(1,3-dioxolan-2-yl)phenol
2973-80-02-BROMO-5-HYDROXYBENZALDEHYDE
■利奥西呱;625115-55-1
625115-55-1Riociguat
51859-98-4(2-fluorobenzyl)hydrazine 
53544-13-1ethyl   3-cyano-2-oxopropanoate  
256504-39-9ethyl   5-amino-1-(2-fluorobenzyl)-1H-pyrazole-3-carboxylate 
256499-19-11-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridine-3-carboximidamide   Hydrochloride
■巴洛沙韦;Baloxavirmarboxil
1985606-14-1Baloxavir   marboxil
119736-16-23-(Benzyloxy)-4-oxo-4H-pyran-2-carboxylic   acid
1228258-40-92-(2-aminoethoxy)-1,1-dimethoxyethane
■曲格列汀;Trelagliptin
865759-25-7Trelagliptin
334618-23-4(R)-3-Aminopiperidine   dihydrochloride  
4270-27-36-Chlorouracil 
421552-12-72-(bromomethyl)-4-fluorobenzonitrile  
■西那卡塞;CINACALCET
364782-34-3CINACALCET
779-89-51.   3-(Trifluoromethyl)cinnamic acid
585-50-22.   3-(3-Trifluoromethylphenyl)propionic acid 
78573-45-23.   3-(3-(trifluoromethyl)phenyl)propan-1-ol 
21172-41-84.   3-[3-(Trifluoromethyl)Phenyl]Propionaldehyde 
42882-31-55.   (+/-)1-(1-Naphthyl)ethylamine 
3886-70-26.   (R)-(+)-alpha-(1-Naphthyl)ethylamine
82572-04-17.   (R)-(+)-alpha-(1-Naphthyl)ethylamine hydrochloride
■艾沙佐米;CITRATE
■库潘尼西;Copanlisib
1032568-63-0Copanlisib
3167-50-82-Aminopyrimidine-5-carboxylic   acid 
2450-26-24-HYDROXY-3-METHOXY-2-NITROBENZALDEHYDE 
887202-50-83-(benzyloxy)-6-(4,5-dihydro-1H-imidazol-2-yl)-2-methoxyaniline 
■维拉佐酮;Vilazodone
163521-12-8Vilazodone 
15861-24-25-Cyanoindole 
143612-79-73-(4-chloro-butyl)-5-cyanoindole  
183288-47-35-(1-piperazinyl)benzofuran-2-carboxylic   acid  
163521-20-85-(1-piperazinyl)benzofuran-2-carboxylic   acid ethyl ester
1422956-31-75-(1-piperazinyl)-2-Benzofurancarboxylic   acid ethyl ester dihydrochloride 
183288-46-25-(1-Piperazinyl)benzofuran-2-carboxamide 
■罗氟司特;Roflumilast
162401-32-3Roflumilast
162401-62-93-Cyclopropylmethoxy-4-difluoromethoxy-benzoic   acid
■伐伦克林;Varenicline
■纳诺醇醚;Oxalate
■瑞卡帕布;Rucaparib
■纳比隆中间体;Nabilone
■培哚普利;Perindoprilat
■维拉帕尼;Veliparib